平安! 发表于 2011-11-9 19:57 @ W# g* J3 h. W/ h; K
Pazopanib (100 mg/kg/day free base equivalent) " `# G5 j- T+ q W
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。- _! G6 J' a9 R; [8 b) _ z& N2 A
搜索了一下,原料一大堆。1 @* g% u) D" f g6 p
: o. P. z; A: r- u+ r, Z对不起!100mg/kg是用于移植瘤的,我弄错了。7 X+ R8 {$ k' p, \& c
$ F0 a: g! Q1 W0 n以下是正版说明书的推荐用量。+ V {& T5 G) ^5 v$ x1 k4 X- J( w& k
7 i9 j- @ ?9 E& D--------------------- DOSAGE AND ADMINISTRATION ----------------
% z( b; \$ t: A$ U- g; l* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
/ ]+ ^3 d3 @6 @' U* r" ^* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) - j3 W5 A% V/ ^
---------------------DOSAGE FORMS AND STRENGTHS --------------1 T4 _8 R5 x1 K
200 mg tablets. (3)
, h+ \* `/ O( j3 @ p- q-------------------------------CONTRAINDICATIONS------------------------ |